Antimo Gioiello

Antimo Gioiello

Università degli Studi di Perugia - Perugia / Italy
Medical and Health Sciences / Pharmacy & Pharmaceutical Sciences
AD Scientific Index ID: 1751967
University of Perugia
person_outline Antimo Gioiello's MOST POPULAR ARTICLES
1-) TGR5-mediated bile acid sensing controls glucose homeostasisC Thomas, A Gioiello, L Noriega, A Strehle, J Oury, G Rizzo, ...Cell metabolism 10 (3), 167-177, 200916362009
2-) TGR5 activation inhibits atherosclerosis by reducing macrophage inflammation and lipid loadingTWH Pols, M Nomura, T Harach, G Lo Sasso, MH Oosterveer, C Thomas, ...Cell metabolism 14 (6), 747-757, 20114772011
3-) Novel potent and selective bile acid derivatives as TGR5 agonists: biological screening, structure− activity relationships, and molecular modeling studiesH Sato, A Macchiarulo, C Thomas, A Gioiello, M Une, AF Hofmann, ...Journal of medicinal chemistry 51 (6), 1831-1841, 20083012008
4-) Discovery of 6α-ethyl-23 (S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesityR Pellicciari, A Gioiello, A Macchiarulo, C Thomas, E Rosatelli, B Natalini, ...Journal of medicinal chemistry 52 (24), 7958-7961, 20092742009
5-) Bile acid derivatives as ligands of the farnesoid X receptor. Synthesis, evaluation, and structure-activity relationship of a series of body and side chain modified analogues …R Pellicciari, G Costantino, E Camaioni, BM Sadeghpour, A Entrena, ...Journal of medicinal chemistry 47 (18), 4559-4569, 20042502004